Class of pharmacological agents, which reduces or diminishes the effect of an agonist on a receptor.
1
The selective δ-opioid receptor antagonist naltrindole only partially blocked the effect of MMP-2200.
2
This effect was blocked only by the kappa-opioid receptor antagonist nor-BNI.
3
These effects of HC were significantly reversed by the glucocorticoid receptor antagonist RU486.
4
Another group received the thrombin receptor antagonist in combination with the standard anti-platelet treatments.
5
These changes were completely prevented by the AII receptor antagonist.
6
The analgesic effects of ASP8062 were significantly blocked by a GABA B receptor antagonist.
7
This effect was blocked by the progesterone receptor antagonist, RU486.
8
Conclusion: Endothelin receptor antagonist and angiotensin II receptor antagonist could prevent against the Nit tolerance.
9
Neither GH secretagogue receptor antagonist nor ghrelin affected the profiles of the insulin tolerance test.
10
Irbesartan is an angiotensin II receptor antagonist indicated for the treatment of patients with hypertension.
11
A significant reduction in clinically important gastrointestinal hemorrhage is evident only with histamine-2- receptor antagonist therapy.
12
Plasma levels of high-sensitivity C-reactive protein and interleukin-1 receptor antagonist were measured in all patients.
13
D2 receptor antagonist triggered arc expression when administered alone.
14
One of these is the endothelin receptor antagonist bosentan.
15
Small scale studies have shown the benzodiazepine receptor antagonist flumazenil to be effective in ameliorating PSE.
16
Furthermore, the extent of protection was comparable to that produced by the NMDA receptor antagonist AP5.