Значения термина full agonist на английском

The full agonist norepinephrine evoked similar FRET changes for all three constructs.

In functional in vitro cation flux assays, A-85380 is a potent and full agonist.

However, the compounds presented here display partial agonist or antagonist behavior instead of full agonist.

Noradrenaline behaved as a full agonist and St-587 as a partial agonist for this response.

Lorazepam is a BZ receptor full agonist and has been used to treat both anxiety and insomnia.

Furthermore, ZK 756326 was a full agonist of CCR8, dose-responsively eliciting an increase in intracellular calcium and cross-desensitizing the response of the receptor to CCL1.

Noradrenaline and St-587 behaved as full agonists inducing a concentration-dependent vasoconstriction.

Moreover, some full agonists became only partial agonists when applied to the S275A receptor.

Key results: All six tested δ receptor agonists were full agonists in the cAMP assay but displayed distinct β-arrestin 2 recruitment efficacy.

Ultimately, as a long-term goal, X-ray crystallography of unoccupied receptors and receptors liganded by partial or full agonists may provide definitive insights.

Not all cannabimetics are bad - technically, paracetamol is one - but the ones sprayed on herbs are full agonists for the receptors.