Class of pharmacological agents, which reduces or diminishes the effect of an agonist on a receptor.
Sinônimos
Examples for "antagonist"
Examples for "antagonist"
1Conclusion: Switching of the TNF antagonist over time is a common issue.
2However, recent analyses of antagonist-occupied receptor function suggest a more complex picture.
3General Saterges had found in Stephen Cordier a powerful antagonist in action.
4Similar effects were observed when microglia were treated with LRP1 antagonist RAP.
5Orexin antagonist leads to significant reduction of sympathetic over-activity during withdrawal syndrome.
1These doses were associated with well-defined pharmacological effects compatible with N-methyl-D-aspartate receptor antagonism.
2Endothelin- receptor antagonism with oral bosentan is an effective approach to therapy for pulmonary arterial hypertension.
3These results emphasize that ET receptor antagonism may yield different results in healthy and diseased states.
4Insulin receptor antagonism increased pancreatic β-cell mass threefold.
5Endothelin (ET) receptor antagonism is a potential therapeutic intervention in the treatment of vascular diseases.
1The selective δ-opioid receptor antagonist naltrindole only partially blocked the effect of MMP-2200.
2This effect was blocked only by the kappa-opioid receptor antagonist nor-BNI.
3These effects of HC were significantly reversed by the glucocorticoid receptor antagonist RU486.
4Another group received the thrombin receptor antagonist in combination with the standard anti-platelet treatments.
5These changes were completely prevented by the AII receptor antagonist.
6The analgesic effects of ASP8062 were significantly blocked by a GABA B receptor antagonist.
7This effect was blocked by the progesterone receptor antagonist, RU486.
8Conclusion: Endothelin receptor antagonist and angiotensin II receptor antagonist could prevent against the Nit tolerance.
9Neither GH secretagogue receptor antagonist nor ghrelin affected the profiles of the insulin tolerance test.
10Irbesartan is an angiotensin II receptor antagonist indicated for the treatment of patients with hypertension.
11A significant reduction in clinically important gastrointestinal hemorrhage is evident only with histamine-2- receptor antagonist therapy.
12Plasma levels of high-sensitivity C-reactive protein and interleukin-1 receptor antagonist were measured in all patients.
13D2 receptor antagonist triggered arc expression when administered alone.
14One of these is the endothelin receptor antagonist bosentan.
15Small scale studies have shown the benzodiazepine receptor antagonist flumazenil to be effective in ameliorating PSE.
16Furthermore, the extent of protection was comparable to that produced by the NMDA receptor antagonist AP5.
Translations for receptor antagonist